One-pot Synthesis of Polysubstituted Indolizine Derivatives
نویسندگان
چکیده مقاله:
An efficient approach to the synthesis of 1,2,3-trisubstituted indolizines is described via one-pot reactions of pyridine and dialkyl acetylendicarboxylate in the presence of ethyl 2-chloroacetoacetate in MeOH at room temperature. The corresponding 1, 2, 3-trisubstituted indolizines may be useful building blocks for the construction of complex indolizine derivatives.
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عنوان ژورنال
دوره 10 شماره 3
صفحات 85- 90
تاریخ انتشار 2016-08-01
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